Compile Data Set for Download or QSAR
maximum 50k data

Found 18 hits with non-zero ITC data for monomer = 517   

CellHIV-1 Protease B Subtype(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -53.1kJ/mole −TΔS°: -61.9kJ/mole ΔH°: 8.78kJ/mole logk: 2.08E+9
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -53.1kJ/mole −TΔS°: -61.9kJ/mole ΔH°: 8.78kJ/mole logk: 2.08E+9
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -51.8kJ/mole −TΔS°: -59.4kJ/mole ΔH°: 7.52kJ/mole logk: 1.30E+9
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant (M46I/I54V)(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -51.0kJ/mole −TΔS°: -65.7kJ/mole ΔH°: 14.6kJ/mole logk: 8.90E+8
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease C Subtype(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -50.6kJ/mole −TΔS°: -60.6kJ/mole ΔH°: 10.0kJ/mole logk: 7.09E+8
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, A-1(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -49.7kJ/mole −TΔS°: -64.8kJ/mole ΔH°: 15.0kJ/mole logk: 5.56E+8
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -49.3kJ/mole −TΔS°: -65.7kJ/mole ΔH°: 16.3kJ/mole
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant (L10I/L90M)(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -49.3kJ/mole −TΔS°: -61.9kJ/mole ΔH°: 12.5kJ/mole logk: 4.30E+8
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease A Subtype(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -48.5kJ/mole −TΔS°: -59.4kJ/mole ΔH°: 10.9kJ/mole logk: 3.13E+8
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant (V82A/I84V)(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -45.1kJ/mole −TΔS°: -60.6kJ/mole ΔH°: 15.5kJ/mole logk: 8.50E+7
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, MDR-QM(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -43.5kJ/mole −TΔS°: -70.3kJ/mole ΔH°: 26.8kJ/mole logk: 4.50E+7
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease B Subtype Mutant (V82F/I84V)(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -42.6kJ/mole −TΔS°: -57.3kJ/mole ΔH°: 14.6kJ/mole logk: 3.13E+7
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease C Subtype Mutant (V82F/I84V)(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -39.7kJ/mole −TΔS°: -52.7kJ/mole ΔH°: 13.0kJ/mole logk: 1.00E+7
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, MDR-HM(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -38.9kJ/mole −TΔS°: -74.0kJ/mole ΔH°: 35.1kJ/mole logk: 6.50E+6
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease A Subtype Mutant (V82F/I84V)(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -38.5kJ/mole −TΔS°: -50.6kJ/mole ΔH°: 12.1kJ/mole logk: 5.20E+6
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant (V82F/I84V)(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -38.5kJ/mole −TΔS°: -63.1kJ/mole ΔH°: 24.7kJ/mole
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, NAM-10(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -35.7kJ/mole −TΔS°: -61.5kJ/mole ΔH°: 25.7kJ/mole logk: 1.86E+6
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, ANAM-11(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
ITC DataΔG°: -32.6kJ/mole −TΔS°: -56.1kJ/mole ΔH°: 23.4kJ/mole logk: 5.26E+5
pH: 5.0 T: 25.00°C 
  • Reorder this table by ΔH°
  • Reorder this table by ΔS°
  • Reorder this table by pH
  • Reorder this table by T
  • Change energy unit to:  kcal/mol