Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ec50 for drug = Fibricor
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28803(2-[4-(4-chlorophenoxy)phenoxy]propanoic acid | Clo...)
Affinity DataIC50: >9.84E+4nM EC50:  1.16E+4nMpH: 8.0 T: 2°CAssay Description:For hPPAR alpha, percentage inhibition was calculated relative to unlabeled GW2331, which was used as the active site-specific competitive binder. Fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Bristol-Myers Squibb

LigandPNGBDBM28803(2-[4-(4-chlorophenoxy)phenoxy]propanoic acid | Clo...)
Affinity DataEC50:  1.77E+4nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Bristol-Myers Squibb

LigandPNGBDBM28803(2-[4-(4-chlorophenoxy)phenoxy]propanoic acid | Clo...)
Affinity DataEC50:  1.85E+4nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mesocricetus auratus (golden hamster))
Bristol-Myers Squibb

LigandPNGBDBM28803(2-[4-(4-chlorophenoxy)phenoxy]propanoic acid | Clo...)
Affinity DataEC50:  2.87E+4nMAssay Description:EC50 is the concentration of test compounds needed to induce 50% of the maximum luciferase activity in HEK cells transfected with PPAR and Gal4-lucif...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28803(2-[4-(4-chlorophenoxy)phenoxy]propanoic acid | Clo...)
Affinity DataIC50: >9.84E+4nM EC50: >5.00E+4nMpH: 8.0 T: 2°CAssay Description:For PPARgamma, the percentage inhibition was calculated relative to rosiglitazone, which was used as the active site-specific competitive binder. Flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed