Compound Name

SMILES String

CC(=O)NC1CCCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC(=O)NC1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC(=O)NC[C@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

CC(C)(C#N)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC(C)(C)Oc1ccc(NC(=O)c2cnc(N3CC[C@@H](O)C3)c(c2)-c2cncnc2)cc1 |r|

CC(C)(C)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)(O)C1CCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC(C)(O)C1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC(C)(O)C1CN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC(C)(O)C1CN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC(C)(O)Cn1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)(O)c1cc(F)cc(c1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CC(C)(O)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC(C)CN1CCN(CCOc2ccc(cc2-c2cncnc2)C(=O)Nc2ccc(OC(F)(F)F)cc2)CC1

CC(C)c1nc2c(cc(cc2n1C)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)-c1cncnc1

CC(C)c1nc2cc(cc(-c3cncnc3)c2n1C)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1c(C)nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1c(nc2cc(cc(-c3cccnn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F

CC(C)n1c(nc2cc(cc(-c3cccnn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)[C@H](C)O |r|

CC(C)n1c(nc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F

CC(C)n1c(nc2cc(cc(-c3ccnnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F

CC(C)n1c(nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F

CC(C)n1c(nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C1CCOCC1

CC(C)n1c(nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)[C@H](C)O |r|

CC(C)n1c(nc2cc(cc(-c3cnsc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F

CC(C)n1c(nc2cc(cc(-c3cscn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F

CC(C)n1cnc2cc(C(=O)Nc3ccc(OC(F)(F)Cl)cc3)c(F)c(Br)c12

CC(C)n1cnc2cc(cc(-c3cccnn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3ccn(C)n3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3ccnn3C)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3cncc(F)c3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3cncs3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3cnn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3cnsc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3cscn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3n[nH]cc3C#N)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3n[nH]cc3O)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-c3noc(=O)[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(-n3cnc(c3)C3CC3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(Br)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(C(=O)NC3CC3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(cc(C(N)=O)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C)n1cnc2cc(nc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(C1COC1)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CC[C@@H](O)C3)c(c2)-c2cncc(F)c2)cc1 |r|

CC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CC[C@@H](O)C3)c(c2)-c2cncc(c2)C#N)cc1 |r|

CC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CC[C@@H](O)C3)c(c2)-c2cncnc2)cc1 |r|

CC1(CC1)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC1(O)CCN(C1)c1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC1(O)CCN(C1)c1ccc(cc1-c1cncs1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC1(O)CCN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC1(O)CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC1(O)CN(C1)c1ncc(cc1-c1[nH]ncc1F)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC1(O)CN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC1(O)CN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CC1(O)CN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC1(O)CN(C1)c1ncc(cc1-c1cnc(Cl)c(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC1(O)CN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC1(O)CN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC1(O)CN(C1)c1ncc(cc1-c1ncc[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC1=[N](C)c2cc(cc(c2N1)-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |c:1|

CCN(CCO)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CCN(CCO)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CCN(CCO)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(SC(F)(F)F)cc1

CCN(CCO)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CCN(CCO)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CCN(CCO)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(SC(F)(F)F)cc1

CCN(CCO)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CCN(CCO)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)F)cc1

CCN(CCO)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(SC(F)(F)F)cc1

CCN(CCO)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CCN(CCO)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CCN(CCO)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(SC(F)(F)F)cc1

CCOc1nc2cc(cc(-c3cncnc3)c2n1C(C)C)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CCOc1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CC[C@@H]1COCc2nc3cc(cc(-c4ccn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

CCc1ccc(cn1)-c1cc(cnc1N1CC[C@H](CO)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CCn1c(CO)nc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CCn1c(OC)nc2cc(cc(-c3cccnn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CCn1c(OC)nc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CCn1c(OC)nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CCn1c(nc2cc(cc(-c3cccnn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F

CCn1c(nc2cc(cc(-c3cccnn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)[C@H](C)O |r|

CCn1c(nc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)[C@@H](C)O |r|

CCn1c(nc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)[C@H](C)O |r|

CCn1c(nc2cc(cc(-c3ccnnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F

CCn1c(nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)[C@H](C)O |r|

CCn1c(nc2cc(cc(-c3cnoc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)[C@H](C)O |r|

CCn1cnc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CN(C)C(=O)c1ccc([nH]1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

CN(C)C1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(C)C1CN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CN(C)C1CN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(C)C1CN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(C)C1CN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(C)CCCN(C)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(C)[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

CN(C)[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CN(C)[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

CN(C)[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CN(C1CCOCC1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(CCCO)c1ncc(cc1-c1ccc(C)nc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(CCCO)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(CCCO)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(CCO)c1ccc(cc1-c1cncs1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(CCO)c1ncc(cc1-c1ccc(C)nc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(CCO)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(CCO)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CN(CCO)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(CCO)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(SC(F)(F)F)cc1

CN(CCO)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CN(CCO)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(CCO)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(SC(F)(F)F)cc1

CN(CCO)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CN(CCO)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(CCO)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(SC(F)(F)F)cc1

CN(CCO)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

CN(CCO)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN(CCO)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(SC(F)(F)F)cc1

CN1CC2CN(CC2C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN1CCCN(CC1)c1ncc(cc1-c1ccc(C)nc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN1CCCN(CC1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN1CCN(CC1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CN[C@@H]1CCN(C1)c1ncc(cc1-c1ccc(C)nc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CN[C@@H]1CCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CN[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CN[C@H]1CCN(C1)c1ncc(cc1-c1ccc(C)nc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CN[C@H]1CCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CN[C@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CNc1c(Br)cc(cc1NC(=O)CC(=O)OC)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

COC(=O)c1cc(Br)c(NCC2(CC2)O[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)c(c1)[N+]([O-])=O

COC(=O)c1cc(F)cc(c1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

COC(=O)c1cc(cs1)-c1cccc(c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COC(=O)c1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COC(OC)OCC(C)(C)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)OC

COCCOc1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COCCOc1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COC[C@@H](C)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

COC[C@H](C)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

CO[C@@H]1CN(C[C@H]1O)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CO[C@H]1CN(C[C@@H]1N)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

CO[C@H]1CN(C[C@@H]1N)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CO[C@H]1CN(C[C@@H]1N)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

CO[C@H]1CN(C[C@@H]1N)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CO[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1cncs1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

CO[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

COc1ccc(CNc2cc(cc3ncn(C(C)C)c23)C(=O)Nc2ccc(OC(F)(F)Cl)cc2)cc1

COc1ccc(Cn2ncc(F)c2-c2cc(cc3ncn(C(C)C)c23)C(=O)Nc2ccc(OC(F)(F)Cl)cc2)cc1 |(-19.35,12.09,;-17.9,11.09,;-18.03,9.34,;-16.58,8.35,;-16.72,6.59,;-18.3,5.83,;-18.44,4.08,;-16.98,3.08,;-15.16,3.39,;-14.26,2.14,;-15.16,.9,;-14.77,-.59,;-16.63,1.37,;-18.69,.24,;-20.02,1.01,;-21.35,.24,;-21.35,-1.3,;-20.02,-2.07,;-19.7,-3.58,;-18.17,-3.74,;-17.54,-2.33,;-16.05,-1.93,;-14.96,-3.02,;-15.65,-.44,;-18.69,-1.3,;-22.69,1.01,;-22.69,2.55,;-24.02,.24,;-25.35,1.01,;-25.35,2.55,;-26.69,3.32,;-28.02,2.55,;-29.35,3.32,;-30.69,2.55,;-32.02,3.32,;-30.69,1.01,;-32.02,1.78,;-28.02,1.01,;-26.69,.24,;-19.76,6.82,;-19.62,8.58,)|

COc1ccc(Cn2ncc(F)c2-c2cc(cc3ncn(C4CC4)c23)C(=O)Nc2ccc(OC(F)(F)Cl)cc2)cc1 |(-15.22,21.52,;-13.88,20.58,;-14.02,18.94,;-12.67,18,;-12.81,16.37,;-14.29,15.67,;-14.43,14.03,;-13.09,13.09,;-11.41,13.47,;-10.5,12.23,;-11.41,10.98,;-11.01,9.49,;-12.87,11.46,;-14.2,10.69,;-15.54,11.46,;-16.87,10.69,;-16.87,9.15,;-15.54,8.38,;-15.22,6.87,;-13.69,6.71,;-13.06,8.12,;-11.57,8.51,;-10.08,8.12,;-10.32,9.77,;-14.2,9.15,;-18.21,11.46,;-18.21,13,;-19.54,10.69,;-20.87,11.46,;-20.87,13,;-22.21,13.77,;-23.54,13,;-24.87,13.77,;-26.21,13,;-27.54,13.77,;-26.21,11.46,;-27.54,12.23,;-23.54,11.46,;-22.21,10.69,;-15.64,16.61,;-15.5,18.24,)|

COc1ccc(cc1-c1cc[nH]n1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ccc(cc1-c1ccc(F)nc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ccc(cc1-c1ccc(s1)C(C)=O)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ccc(cc1-c1ccc2OCOc2c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ccc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ccc(cc1-c1ccncc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ccc(cn1)-c1cc(cnc1N1CC[C@@H](CN)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

COc1ccc(cn1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

COc1ccc(cn1)-c1cc(cnc1NCCCO)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1cncc(c1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

COc1nc2cc(cc(-c3cccnn3)c2n1[C@H](C)CO)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

COc1nc2cc(cc(-c3ccn[nH]3)c2n1C(C)C)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

COc1nc2cc(cc(-c3ccn[nH]3)c2n1[C@H](C)CO)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

COc1nc2cc(cc(-c3cncnc3)c2n1C(C)C)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

COc1nc2cc(cc(-c3cncnc3)c2n1[C@H](C)CO)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

COc1ncc(c(OC)n1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

COc1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ncc(cc1C#N)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

COc1ncc(cn1)-c1cc(cc2ncn(C(C)C)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

COc1ncc(cn1)-c1cc(cc2ncn(C3CC3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

COc1ncc(cn1)-c1cc(ccc1C)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ncc(cn1)-c1cc(ccc1Cl)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ncc(cn1)-c1cc(ccc1F)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ncc(cn1)-c1cc(ccc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

COc1ncc(cn1)-c1cc(ccn1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ncc(cn1)-c1cc(cnc1N1CCC(O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

COc1ncc(cn1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

COc1ncccc1-c1cncc(c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

CS(=O)(=O)c1ccc(cc1)-c1cnc(NCc2ccco2)n2cnnc12

CSc1nc2cc(cc(Br)c2n1[C@@H](C)[C@H](O)CO)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H](C(F)F)n1cnc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H](C(F)F)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H](C1CC1)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H](CC#N)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H](CF)n1c(nc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F |r|

C[C@@H](CF)n1c(nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F |r|

C[C@@H](CF)n1cnc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H](CF)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H](CO)n1cnc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H](CO)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H](O)Cn1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H](O)c1nc2cc(cc(-c3ccn[nH]3)c2n1C(C)C)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCOc2nc3cc(cc(-c4[nH]ncc4F)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCOc2nc3cc(cc(-c4cccnn4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCOc2nc3cc(cc(-c4ccn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCOc2nc3cc(cc(-c4ccnnc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCOc2nc3cc(cc(-c4cncc(c4)C#N)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCOc2nc3cc(cc(-c4cncnc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCOc2nc3cc(cc(-c4cnoc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCOc2nc3cc(cc(-c4cnsc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCOc2nc3cc(cc(-c4cscn4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCSc2nc3cc(cc(-c4ccn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCSc2nc3cc(cc(-c4cncnc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1CCc2nc3cc(cc(-c4ccn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4[nH]ncc4C#N)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4[nH]ncc4C)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4[nH]ncc4F)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4cc(O)ccn4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

C[C@@H]1COCc2nc3cc(cc(-c4cc(n[nH]4)C#N)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4cc(n[nH]4)C4CC4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4cccnn4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4ccn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4ccn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4ccnnc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4cncc(c4)C#N)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4cncnc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4cncnc4)c3n12)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4cncs4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4cnn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4cnoc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4cnsc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4csc(C)n4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4csc(n4)C#N)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4cscn4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4ncco4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(-c4nccs4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(Br)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COCc2nc3cc(cc(N4CCC4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1COc2nc3cc(cc(-c4cccnn4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

C[C@@H]1COc2nc3cc(cc(-c4ccn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

C[C@@H]1CSc2nc3cc(cc(-c4ccn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1C[C@H]1n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1Cn2c(CO1)nc1cc(cc(-c3cncnc3)c21)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@H]1[C@H](O)COc2nc3cc(cc(-c4ccn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@]1(O)CCN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@@]1(O)CCN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

C[C@@]1(O)CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

C[C@H](C(F)F)n1cnc2cc(cc(-c3cccnn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](C(F)F)n1cnc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](C(F)F)n1cnc2cc(cc(-c3ccnnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](C(F)F)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](C1CC1)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](CC#N)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](CF)n1c(nc2cc(cc(-c3cccnn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F |r|

C[C@H](CF)n1c(nc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F

C[C@H](CF)n1c(nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F |r|

C[C@H](CF)n1cnc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](CF)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](CO)n1c(C)nc2cc(cc(-c3cccnn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](CO)n1c(C)nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](CO)n1c(nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F

C[C@H](CO)n1cnc2cc(cc(-c3cccnn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](CO)n1cnc2cc(cc(-c3ccn[nH]3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](CO)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](O)Cn1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H](O)c1nc2cc(cc(-c3ccn[nH]3)c2n1C(C)C)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

C[C@H](n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(C)(C)O |r|

C[C@H]1COCc2nc3cc(cc(-c4cncnc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H]1Cn2c(CO1)nc1cc(cc(-c3cncnc3)c21)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@H]1OCC[C@H]1n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@]1(O)CCCN(C1)c1c(Br)cc(cc1[N+]([O-])=O)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@]1(O)CCN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

C[C@]1(O)CCN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

C[C@]1(O)CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1cc([nH]n1)-c1cc(ccc1N1C[C@H](N)[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

Cc1cc([nH]n1)-c1cc(cnc1N1CC(C)(O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

Cc1cc([nH]n1)-c1cc(cnc1N1CC(CO)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

Cc1cc([nH]n1)-c1cc(cnc1N1CC(CO)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1cc([nH]n1)-c1cc(cnc1N1CC(O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

Cc1cc([nH]n1)-c1cc(cnc1N1CC(O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(F)cc1-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

Cc1ccc(F)cc1-c1cc(cnc1N1C[C@H](O)[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

Cc1ccc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cc1-c1cncs1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cc1-n1ccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cn1)-c1cc(ccc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(ccc1N1C[C@H](O)[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1N1CC(C)(O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cn1)-c1cc(cnc1N1CC(C1)C(C)(C)O)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cn1)-c1cc(cnc1N1CC(CO)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cn1)-c1cc(cnc1N1CC(O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cn1)-c1cc(cnc1N1CCC(C1)C(C)(C)O)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cn1)-c1cc(cnc1N1CCC(O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cn1)-c1cc(cnc1N1CCCC(O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cn1)-c1cc(cnc1N1CCC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1N1CCC[C@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1N1CC[C@@H](CN)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1N1CC[C@@H](CO)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1N1CC[C@@H](N)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)C(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1N1CC[C@H](CN)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1N1CC[C@H](CO)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1N1CC[C@H](N)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1N1CC[C@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ccc(cn1)-c1cc(cnc1NCCCO)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccc(cn1)-c1cc(cnc1NCCO)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ccncc1-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

Cc1cnc([nH]1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1cncc(c1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1nc2c(cc(cc2n1C)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)-c1cncc(F)c1

Cc1nc2c(cc(cc2n1C)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)-c1cncnc1

Cc1nc2cc(cc(-c3cncnc3)c2n1C)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

Cc1nc2cc(cc(-c3cncnc3)c2n1C1CC1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

Cc1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ncc(cc1F)-c1cc(cnc1N1CC(C)(O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ncc(cc1F)-c1cc(cnc1N1CC(CO)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ncc(cc1F)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ncc(cc1F)-c1cc(cnc1N1CC[C@H](CO)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ncc(cn1)-c1cc(ccc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ncc(cn1)-c1cc(ccc1N1C[C@H](O)[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

Cc1ncc(cn1)-c1cc(cnc1N1CC(C)(O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ncc(cn1)-c1cc(cnc1N1CC(CO)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cc1ncc(cn1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ncc(cn1)-c1cc(cnc1N1CC[C@H](CO)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ncc(cn1)-c1cc(cnc1N1C[C@H](O)[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

Cc1ncc(s1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ncc(s1)-c1cc(cnc1N1CC[C@H](CO)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ncccc1-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

Cc1ncccc1-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Cc1ncncc1-c1cc(ccc1N1C[C@H](O)[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

Cc1ncncc1-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

Cc1ncncc1-c1cc(cnc1N1C[C@@H](O)[C@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

Cn1c(CO)nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

Cn1c(ccc1-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C#N |r|

Cn1c(nc2c(cc(cc12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)-c1cncnc1)C(F)F

Cn1c(nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(C)(C)O

Cn1c(nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)F

Cn1c(nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C1CC1

Cn1c(nc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C1CCC1

Cn1cc(cn1)-c1cc(ccc1Cl)C(=O)Nc1ccc(OC(F)(F)F)cc1

Cn1cc(cn1)-c1cc(ccc1F)C(=O)Nc1ccc(OC(F)(F)F)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3ccn[nH]3)c3n(cnc3c2)C2CC2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3ccn[nH]3)c3n4CCOCc4nc3c2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3[nH]cnc3c2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(CC4CC4)cnc3c2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(CC4COC4)cnc3c2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(C[C@@H]4CCCO4)cnc3c2)cc1 |r|

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(C[C@H]4CCCO4)cnc3c2)cc1 |r|

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(cnc3c2)C2CC(F)(F)C2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(cnc3c2)C2CC2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(cnc3c2)C2CCC2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(cnc3c2)C2CCCC2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(cnc3c2)C2CCOC2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(cnc3c2)C2CS(=O)(=O)C2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(cnc3c2)[C@@H]2CCOC2)cc1 |r|

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(cnc3c2)[C@@H]2CNC(=O)C2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(cnc3c2)[C@H]2CCOC2)cc1 |r|

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(-c3cncnc3)c3n(cnc3c2)[C@H]2CNC(=O)C2)cc1 |r|

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(Br)c3n(CC(=O)NC4CC4)cnc3c2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(Br)c3n4CCCCc4nc3c2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cc(Br)c3n4CCS(=O)(=O)Cc4nc3c2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cccc(c2)-c2cncnc2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(Cl)c(c2)-c2cncnc2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(N3CC4(CNC4)C3)c(c2)-c2ccn[nH]2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(N3CCC(F)(F)C3)c(c2)-c2ccn[nH]2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(N3CCC(F)(F)C3)c(c2)-c2cncnc2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(N3CCC4(CNC4)C3)c(c2)-c2ccn[nH]2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(N3CCCC4(CCN4)C3)c(c2)-c2ccn[nH]2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(N3CCN(CC3)C3CC3)c(c2)-c2ccn[nH]2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(N3CCNC4(CC4)C3)c(c2)-c2ccn[nH]2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(N3CCNC4(CC4)C3)c(c2)-c2cncnc2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(N3CCOCC3)c(c2)-c2ccn[nH]2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(N3Cc4cn[nH]c4C3)c(c2)-c2cncnc2)cc1

FC(F)(Cl)Oc1ccc(NC(=O)c2cnc(OC3CCOCC3)c(c2)-c2cncnc2)cc1

FC(F)(F)CN1CCN(CC1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

FC(F)(F)Cc1ccc(NC(=O)c2cccc(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cc(ccn2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2ccc(Cl)c(c2)-c2cc[nH]n2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2ccc(Cl)c(c2)-c2cccnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2ccc(Cl)c(c2)-c2ccncc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2ccc(Cl)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2ccc(N3CCOC3=O)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2ccc(OCCN3CCCC3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2ccc(OCCN3CCOCC3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cccc(c2)-c2ccc(CN3CCCC3)s2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cccc(c2)-c2cncc(c2)C#N)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cccc(c2)-c2cnccn2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cccc(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cccc(c2)-n2ccnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cccc(n2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2ccnc(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(C3=CCOCC3)c(c2)-c2cncnc2)cc1 |t:16|

FC(F)(F)Oc1ccc(NC(=O)c2cnc(C3CCOCC3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(Cl)c(c2)-c2cccnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(Cl)c(c2)-c2ccn[nH]2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(Cl)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(Cl)c(c2)-c2ncc[nH]2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3C4COCC3COC4)c(c2)-c2cncnc2)cc1 |TLB:15:16:22.23.24:18.20.19|

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCC(F)(F)C3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCC4(CCNC4=O)C3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCC4(COC4)C3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCCC3)c(c2)-c2cc(n[nH]2)C#N)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCCC3)c(c2)-c2ccn[nH]2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCCC3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCCNCC3)c(c2)-c2cccnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCCOCC3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCC[C@@H](C3)C#N)c(c2)-c2cncnc2)cc1 |r|

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCC[C@H](C3)C#N)c(c2)-c2cncnc2)cc1 |r|

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCNC4(CC4)C3)c(c2)-c2ccn[nH]2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCNC4(CC4)C3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCOCC3)c(c2)-c2ccn[nH]2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3CCOCC3)c(c2)-c2cnccn2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3Cc4ccncc4C3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(N3Cc4cn[nH]c4C3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(OC3CCOCC3)c(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(c(c2)-c2cncnc2)C(F)(F)F)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(c(c2)-c2cncnc2)C2(CCC2)C#N)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cnc(c(c2)-c2cncnc2)C2(CCOCC2)C#N)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cncc(c2)-c2cccnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cncc(c2)-c2cncnc2)cc1

FC(F)(F)Oc1ccc(NC(=O)c2cncc(n2)-c2cncnc2)cc1

FC(F)(F)Sc1ccc(NC(=O)c2cccc(c2)-c2cncnc2)cc1

FC(F)CN1CCN(CC1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

FC(F)Cn1cnc2cc(cc(-c3cccnn3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

FC(F)Cn1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

FC(F)c1nc2cc(cc(-c3ccn[nH]3)c2n1C1CC1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

FC(F)c1nc2cc(cc(Br)c2n1C1CC1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

FCCN1CCN(CC1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

FC[C@@H]1COCc2nc3cc(cc(Br)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

F[C@H]1C[C@@H](C1)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r,wU:3.5,wD:1.0,(9.78,-.76,;8.29,-1.16,;6.96,-.39,;6.19,-1.72,;7.52,-2.49,;4.7,-2.12,;4.07,-3.53,;2.54,-3.37,;2.22,-1.86,;.89,-1.09,;.89,.45,;2.22,1.22,;3.56,.45,;4.89,1.22,;6.22,.45,;7.56,1.22,;7.56,2.76,;6.22,3.53,;4.89,2.76,;3.56,-1.09,;-.44,1.22,;-.44,2.76,;-1.78,.45,;-3.11,1.22,;-4.45,.45,;-5.78,1.22,;-5.78,2.76,;-7.11,3.53,;-8.45,2.76,;-9.78,3.53,;-8.45,1.22,;-9.78,1.99,;-4.45,3.53,;-3.11,2.76,)|

F[C@H]1C[C@H](C1)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r,wU:3.5,1.0,(9.78,-.76,;8.29,-1.16,;7.52,-2.49,;6.19,-1.72,;6.96,-.39,;4.7,-2.12,;4.07,-3.53,;2.54,-3.37,;2.22,-1.86,;.89,-1.09,;.89,.45,;2.22,1.22,;3.56,.45,;4.89,1.22,;6.22,.45,;7.56,1.22,;7.56,2.76,;6.22,3.53,;4.89,2.76,;3.56,-1.09,;-.44,1.22,;-.44,2.76,;-1.78,.45,;-3.11,1.22,;-4.45,.45,;-5.78,1.22,;-5.78,2.76,;-7.11,3.53,;-8.45,2.76,;-9.78,3.53,;-8.45,1.22,;-9.78,1.99,;-4.45,3.53,;-3.11,2.76,)|

Fc1c(cccc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Fc1cc(NC(=O)c2cccc(c2)-c2cncnc2)ccc1OC(F)(F)F

Fc1ccc(cc1-c1cc[nH]n1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Fc1ccc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Fc1ccc(cc1-c1ccncc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Fc1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Fc1ccc(cc1C(=O)Nc1ccc(OC(F)(F)F)cc1)-c1cncnc1

Fc1cncc(c1)-c1cc(cc2ncn(C3CC3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

Fc1cncc(c1)-c1cc(cnc1Cl)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

Fc1cncc(c1)-c1cc(cnc1Cl)C(=O)Nc1ccc(OC(F)(F)F)cc1

Fc1cncc(c1)-c1cncc(c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

NC(=O)C1CCN(CC1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

NC12CC1CN(C2)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

NC12CC1CN(C2)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

NC12CC1CN(C2)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

NC12CC1CN(C2)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

NC1CN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

NC1CN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

NC1CN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

NC1CN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

NCC1(F)CCN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

NCC1(O)CCN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

NCC1CN(CC1O)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

NCC1CN(CC1O)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

NC[C@@H]1CCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

NC[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

NC[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

NC[C@H]1CCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

NC[C@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

NC[C@H]1CN(C[C@H]1O)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

N[C@@H]1CCCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

N[C@@H]1CCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

N[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

N[C@@H]1CN(C[C@H]1F)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

N[C@@]1(CCN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1)C(F)(F)F |r|

N[C@@]1(CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(F)(F)F |r|

N[C@@]1(CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1)C(F)(F)F |r|

N[C@H]1CCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

N[C@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

N[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

N[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

N[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

N[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

N[C@H]1[C@@H]2CN(C[C@H]12)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

N[C@H]1[C@@H]2CN(C[C@H]12)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

N[C@H]1[C@@H]2CN(C[C@H]12)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

N[C@H]1[C@@H]2CN(C[C@H]12)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Nc1cnc(cn1)-c1cccc(c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Nc1ncc(cc1F)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

Nc1ncc(cc1F)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Nc1ncc(cn1)-c1cc(cnc1N1CCCC1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Nc1ncc(cn1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

Nc1ncc(cn1)-c1cncc(c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

O.O[C@@H]1CCCn2c1nc1cc(cc(-c3cccnn3)c21)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC(=O)CCNc1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OC(=O)CCNc1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OC(CCNc1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1)C(O)=O

OC1CCCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OC1CCCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OC1CCN(C1)c1ncc(cc1-c1ccc(nc1)C(F)(F)F)C(=O)Nc1ccc(OC(F)(F)F)cc1

OC1CCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OC1CCN(C1)c1ncc(cc1-c1ccncc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OC1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OC1CCN(CC1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OC1CCN(CC1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OC1CN(C1)c1ncc(cc1-c1[nH]ncc1F)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OC1CN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OC1CN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OC1CN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OC1CN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCC(O)CCNc1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OCC1(CC1)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OCC1CCCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCC1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCC1CN(C1)c1ncc(cc1-c1[nH]ncc1F)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OCC1CN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCC1CN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OCC1CN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCC1CN(C1)c1ncc(cc1-c1cnc(Cl)c(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCC1CN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCC1CN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OCC1CN(CCO1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCC1CN(CCO1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCCC(O)CNc1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OCCCNc1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCCCNc1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCCN(CCO)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OCCN1CC2CN(CC2C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCCNCCOc1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCCNc1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCCOc1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCCOc1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCCOc1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCCOc1ncc(cn1)-c1cccc(c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCC[C@@H](O)CNc1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OCC[C@H](O)CNc1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OCC[C@H]1COc2nc3cc(cc(-c4ccn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OCCn1cc(cn1)-c1cncc(c1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OC[C@@H](O)CCNc1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@@H]1CCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@@H]1CCN(C[C@@H]1O)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@@H]1CCOc2nc3cc(cc(-c4cccnn4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OC[C@@H]1CCOc2nc3cc(cc(-c4cncnc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@@H]1COCc2nc3cc(cc(-c4cccnn4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@@H]1COCc2nc3cc(cc(-c4ccn[nH]4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

OC[C@@H]1COCc2nc3cc(cc(-c4ccnnc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@@H]1COCc2nc3cc(cc(-c4cncnc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@@H]1COc2nc3cc(cc(-c4cccnn4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@@H]1COc2nc3cc(cc(-c4cncnc4)c3n12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@H](O)CCNc1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1ccc(CF)nc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1ccc(Cl)nc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1ccc(nc1)C#N)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1ccc(nc1)C1CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cnc(Cl)c(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cnc(nc1)C#N)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)c(F)c1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(SC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)F)c(F)c1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(SC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)c(F)c1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(SC(F)(F)F)cc1 |r|

OC[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1cncs1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OC[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

OC[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cncs1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OCc1cc([nH]n1)-c1cc(cnc1N1CCCC1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCc1cc(cs1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OCc1ccc(cn1)-c1cc(cnc1N1CCCC1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCc1ccc(cn1)-c1cc(cnc1N1CCOCC1)C(=O)Nc1ccc(OC(F)(F)F)cc1

OCc1ccc(cn1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

OCc1cccc(c1)-c1cc(cnc1N1CC[C@@H](O)C1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCC(N1)c1ncc(cc1-c1cc(F)cc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCC1n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCCN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCCn2c1nc1cc(cc(-c3ccn[nH]3)c21)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

O[C@@H]1CCCn2c1nc1cc(cc(-c3cncnc3)c21)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ccc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ccc(cc1-c1cncs1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cc(F)cc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cc(F)ccc1C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cc(F)cnc1C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cc(F)cnc1Cl)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cc(F)cnc1F)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cc(F)cnc1F)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cc(F)nc(F)c1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cc(F)nc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cc(ccc1F)C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccc(F)nc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccc([nH]1)C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccc([nH]1)C#N)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccc(nc1)C(F)(F)F)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccc2ccncc2c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccc2nccnc2c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccc[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccc[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccc[nH]1)C(=O)Nc1ccc(SC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cccc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccccc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccccn1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cccnc1F)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cccnc1F)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ccoc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cnc(Cl)c(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(Cl)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)C(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)C(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)c(F)c1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(SC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(SC(F)(F)F)c(F)c1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(SC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(cc1)C(F)(F)C(F)(F)F |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(cc1)S(=O)C(F)(F)F |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(cc1)S(F)(F)(F)(F)F |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)F)c(F)c1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(SC(F)(F)F)c(F)c1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(SC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(cc1)C(F)(F)C(F)(F)F |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncc(c1)C(F)(F)F)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cnccc1C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cnccc1C#N)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cnccc1F)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cnccc1F)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)C(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)c(Cl)c1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)c(F)c1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(SC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(SC(F)(F)F)c(F)c1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(SC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(SC(F)(F)F)nc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(SC(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(cc1)C(F)(F)C(F)(F)Cl |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(cc1)C(F)(F)C(F)(F)F |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(cc1)S(=O)(=O)C(F)(F)F |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(cc1)S(F)(F)(F)(F)F |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cncs1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1cnoc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ncc[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1ncc[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCN(C1)c1ncc(cc1-c1nccs1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@@H]1CCc2nc3cc(cc(-c4ccn[nH]4)c3n2C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCn2c(C1)nc1cc(cc(-c3cccnn3)c21)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1CCn2c(C1)nc1cc(cc(-c3cncnc3)c21)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1COC[C@@H]1n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@@H]1COc2nc3cc(cc(-c4ccn[nH]4)c3n2C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

O[C@H]1CC(C1)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r,wU:1.0,(10.82,.04,;9.43,-.64,;8.83,-1.88,;7.3,-1.72,;7.93,-.32,;5.81,-2.12,;5.19,-3.53,;3.65,-3.37,;3.33,-1.86,;2,-1.09,;2,.45,;3.33,1.22,;4.67,.45,;6,1.22,;7.34,.45,;8.67,1.22,;8.67,2.76,;7.34,3.53,;6,2.76,;4.67,-1.09,;.67,1.22,;.67,2.76,;-.67,.45,;-2,1.22,;-3.33,.45,;-4.67,1.22,;-4.67,2.76,;-6,3.53,;-7.34,2.76,;-8.67,3.53,;-7.34,1.22,;-8.67,1.99,;-3.33,3.53,;-2,2.76,)|

O[C@H]1CCCN(C1)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CCCN(C1)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CCCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CCCn2c1nc1cc(cc(-c3ccn[nH]3)c21)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CCN(C1)c1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CCN(C1)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(SC(F)(F)F)cc1 |r|

O[C@H]1CCc2nc3cc(cc(-c4cccnn4)c3n2C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CCc2nc3cc(cc(-c4ccn[nH]4)c3n2C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CCc2nc3cc(cc(-c4cncnc4)c3n2C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1

O[C@H]1CCc2nc3cc(cc(-c4cnoc4)c3n2C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CCn2c(C1)nc1cc(cc(-c3cccnn3)c21)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CCn2c(C1)nc1cc(cc(-c3cncnc3)c21)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@@H]1F)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@@H]1F)c1ncc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1ccc([nH]1)C#N)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1ccc[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1ccn[nH]1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ccc(cc1-c1cncs1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1ccc([nH]1)C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1ccc([nH]1)C#N)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cccnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cnccc1C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@@H]1O)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@H]1O)c1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CN(C[C@H]1O)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@H]1O)c1ncc(cc1-c1cncc(F)c1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1CN(C[C@H]1O)c1ncc(cc1-c1cncc(c1)C#N)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@H]1O)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1CN(C[C@H]1O)c1ncc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1 |r|

O[C@H]1COC[C@@H]1n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1COC[C@H]1n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1COc2nc3cc(cc(-c4cccnn4)c3n2C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1COc2nc3cc(cc(-c4ccn[nH]4)c3n2C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1COc2nc3cc(cc(-c4cncnc4)c3n2C1)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r|

O[C@H]1C[C@@H](C1)n1cnc2cc(cc(-c3cncnc3)c12)C(=O)Nc1ccc(OC(F)(F)Cl)cc1 |r,wU:3.5,wD:1.0,(9.78,-.76,;8.29,-1.16,;6.96,-.39,;6.19,-1.72,;7.52,-2.49,;4.7,-2.12,;4.07,-3.53,;2.54,-3.37,;2.22,-1.86,;.89,-1.09,;.89,.45,;2.22,1.22,;3.56,.45,;4.89,1.22,;6.22,.45,;7.56,1.22,;7.56,2.76,;6.22,3.53,;4.89,2.76,;3.56,-1.09,;-.44,1.22,;-.44,2.76,;-1.78,.45,;-3.11,1.22,;-4.45,.45,;-5.78,1.22,;-5.78,2.76,;-7.11,3.53,;-8.45,2.76,;-9.78,3.53,;-8.45,1.22,;-9.78,1.99,;-4.45,3.53,;-3.11,2.76,)|

Oc1ccc(cc1-c1cncnc1)C(=O)Nc1ccc(OC(F)(F)F)cc1

Oc1ncccc1-c1cncc(c1)C(=O)Nc1ccc(OC(F)(F)F)cc1