Found 3 Enz. Inhib. hit(s) with Target = 'Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R224C]'
TargetGamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R224C](Homo sapiens (Human))
University of Wisconsin At Madison
University of Wisconsin At Madison
Affinity DataKi: 3.30nM ΔG°: -48.4kJ/moleT: 2°CAssay Description:Membrane homogenates were incubated at room temperature with a sub-Kd concentration of radioligand in the absence or presence of seven different conc...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R224C](Homo sapiens (Human))
University of Wisconsin At Madison
University of Wisconsin At Madison
Affinity DataKi: 67.4nM ΔG°: -40.9kJ/moleT: 2°CAssay Description:Membrane homogenates were incubated at room temperature with a sub-Kd concentration of radioligand in the absence or presence of seven different conc...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R224C](Homo sapiens (Human))
University of Wisconsin At Madison
University of Wisconsin At Madison
Affinity DataKi: 70.9nM ΔG°: -40.8kJ/moleT: 2°CAssay Description:Membrane homogenates were incubated at room temperature with a sub-Kd concentration of radioligand in the absence or presence of seven different conc...More data for this Ligand-Target Pair