TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 21.7nMAssay Description:Inhibition of human TLK1 using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 30.4nMAssay Description:Inhibition of human TLK1 using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 30.4nMAssay Description:Inhibition of human TLK1 using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 36.4nMAssay Description:Inhibition of human TLK1 using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of TLK1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: <5.00E+3nMAssay Description:Inhibition of human N-terminal FLAG, C-terminal HIS8-tagged TLK1 expressed in sf9 cells by flashplate based radiometric 33pan-quinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant full-length human TLK1 using casein as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintill...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human TLK1 using histone H3 as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of NanoLuc-fused TLK1 (unknown origin) expressed in HEK293T cells after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 630nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 27nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 740nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TLK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding affinity to TLK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 27nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 27nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TLK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TLK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 740nMAssay Description:Binding affinity to TLK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TLK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TLK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 490nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 1.30E+3nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 630nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 1(Homo sapiens (Human))
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKd: 2.70E+3nMAssay Description:Binding constant for TLK1 kinase domainMore data for this Ligand-Target Pair