TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.00650nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0130nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Torpedo californica electric organ synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Binding affinity to VAChTMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Torpedo californica electric organ synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Binding to vesicular acetylcholine transporter of torpedo synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0630nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.121nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]vesamicol from Vesicular Acetylcholine Transporter (VAChT)More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of (-)-[3H]vesamicol from human VAChT expressed in rat PC12 A123.7 cells after 20 hrsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Binding to vesicular acetylcholine transporter of torpedo synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.147nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.212nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Binding affinity to VAChTMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of (-)-[3H]vesamicol from human VAChT expressed in rat PC12 A123.7 cells after 20 hrsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.248nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]vesamicol from Vesicular Acetylcholine Transporter (VAChT)More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.264nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.271nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]vesamicol from Vesicular Acetylcholine Transporter (VAChT)More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.320nMAssay Description:Binding affinity to VAchTMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Torpedo californica electric organ synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.360nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.360nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.360nMAssay Description:Binding to vesicular acetylcholine transporter of torpedo synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.360nMAssay Description:Binding to vesicular acetylcholine transporter of torpedo synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]vesamicol from Vesicular Acetylcholine Transporter (VAChT)More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.440nMAssay Description:Binding to vesicular acetylcholine transporter of torpedo synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.440nMAssay Description:Displacement of [3H]vesamicol from Vesicular Acetylcholine Transporter (VAChT)More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.440nMAssay Description:Binding affinity to VAchTMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.480nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.530nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.540nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.638nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.660nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.660nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.670nMAssay Description:Binding to vesicular acetylcholine transporter of torpedo synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.762nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.770nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.780nMAssay Description:Displacement of (-)-[3H]vesamicol from human VAChT expressed in rat PC12 cell membrane after 20 hrsMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.798nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:In vitro binding affinity to vesamicol receptor using [3H]-vesamicol.More data for this Ligand-Target Pair