Compile Data Set for Download or QSAR
maximum 50k data
Found 16 of Enz. Inhib. data with enzyme = '17-beta-hydroxysteroid dehydrogenase type 2' and Substrate = '[2,4,6,7-3H]-E2'
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25856(3-[4-(3-hydroxyphenyl)thiophen-2-yl]phenol | hydro...)
Affinity DataIC50:  559nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25839(3-[5-(3-hydroxyphenyl)-1,2,4-thiadiazol-3-yl]pheno...)
Affinity DataIC50:  602nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25851(3-[5-(3-hydroxyphenyl)thiophen-2-yl]phenol | hydro...)
Affinity DataIC50:  745nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25855(3-[4-(4-hydroxyphenyl)thiophen-2-yl]phenol | hydro...)
Affinity DataIC50:  1.27E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25853(4-[4-(3-hydroxyphenyl)thiophen-2-yl]phenol | hydro...)
Affinity DataIC50:  1.69E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25850(3-[5-(4-hydroxyphenyl)thiophen-2-yl]phenol | hydro...)
Affinity DataIC50:  1.95E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25838(4-[5-(3-hydroxyphenyl)-1,2,4-thiadiazol-3-yl]pheno...)
Affinity DataIC50:  2.19E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25836(3-[2-(3-hydroxyphenyl)-1,3-thiazol-4-yl]phenol | h...)
Affinity DataIC50:  2.22E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25863(3-[4-(3-hydroxyphenyl)phenyl]phenol | hydroxypheny...)
Affinity DataIC50:  2.26E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25847(3-(5-phenylthiophen-2-yl)phenol | hydroxyphenyl su...)
Affinity DataIC50:  2.34E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25832(3-[2-(3-hydroxyphenyl)-1,3-thiazol-5-yl]phenol | h...)
Affinity DataIC50:  2.50E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25865(3-[5-(3-hydroxyphenyl)pyridin-2-yl]phenol | hydrox...)
Affinity DataIC50:  3.40E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25831(4-[2-(3-hydroxyphenyl)-1,3-thiazol-5-yl]phenol | h...)
Affinity DataIC50:  4.00E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25864(3-[4-(4-hydroxyphenyl)phenyl]phenol | hydroxypheny...)
Affinity DataIC50:  4.51E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25867(3-[6-(3-hydroxyphenyl)-1,2,4,5-tetrazin-3-yl]pheno...)
Affinity DataIC50:  5.10E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target17-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Saarland University

LigandPNGBDBM25866(3-[5-(3-hydroxyphenyl)pyrazin-2-yl]phenol | hydrox...)
Affinity DataIC50:  5.50E+3nMAssay Description:Tritiated E2 was incubated with 17beta-HSD2, cofactor, and inhibitor. The amount of labeled E1 formed was quantified by HPLC. Detection and quantific...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed