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Found 11 of Enz. Inhib. data with enzyme = 'Calpain-1 catalytic subunit' and Substrate = 'BDBM23856'
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
University of Tennessee Health Science Center

LigandPNGBDBM23865(3-[(2S)-2-[1-(9H-fluoren-9-yl)acetamido]-4-methylp...)
Affinity DataKi:  8nM ΔG°:  -10.9kcal/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
University of Tennessee Health Science Center

LigandPNGBDBM23866(MDL28170 | Z-Val-Phe-CHO | benzyl N-[(1S)-2-methyl...)
Affinity DataKi:  10nM ΔG°:  -10.8kcal/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
University of Tennessee Health Science Center

LigandPNGBDBM23859(3-[(2S)-2-[1-(adamantan-1-yl)acetamido]-4-methylpe...)
Affinity DataKi:  41nM ΔG°:  -9.97kcal/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
University of Tennessee Health Science Center

LigandPNGBDBM23857(3-[(2S)-2-(3-cyclohexylpropanamido)-4-methylpentan...)
Affinity DataKi:  50nM ΔG°:  -9.85kcal/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
University of Tennessee Health Science Center

LigandPNGBDBM23863(3-[(2S)-2-(3,3-diphenylpropanamido)-4-methylpentan...)
Affinity DataKi:  63nM ΔG°:  -9.72kcal/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
University of Tennessee Health Science Center

LigandPNGBDBM23861(3-[(2S)-2-(1,1-diphenylacetamido)-4-methylpentanam...)
Affinity DataKi:  108nM ΔG°:  -9.40kcal/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
University of Tennessee Health Science Center

LigandPNGBDBM23858(Peptidyl alpha-Ketoester, 1b | methyl 3-[(2S)-2-[1...)
Affinity DataKi:  450nM ΔG°:  -8.57kcal/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
University of Tennessee Health Science Center

LigandPNGBDBM23860(Peptidyl alpha-Ketoester, 1c | methyl 3-[(2S)-2-(1...)
Affinity DataKi:  944nM ΔG°:  -8.13kcal/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
University of Tennessee Health Science Center

LigandPNGBDBM23855(Peptidyl alpha-Ketoester, 1a | methyl 3-[(2S)-2-(3...)
Affinity DataKi:  1.05E+3nM ΔG°:  -8.07kcal/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
University of Tennessee Health Science Center

LigandPNGBDBM23864(Peptidyl alpha-Ketoester, 1e | methyl 3-[(2S)-2-[1...)
Affinity DataKi:  1.20E+3nM ΔG°:  -7.99kcal/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
University of Tennessee Health Science Center

LigandPNGBDBM23862(Peptidyl alpha-Ketoester, 1d | methyl 3-[(2S)-2-(3...)
Affinity DataKi:  2.15E+3nM ΔG°:  -7.65kcal/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed