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Found 11 of Enz. Inhib. data with enzyme = 'Serine/threonine-protein kinase pim-1' and Substrate = 'BDBM220099'
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM218904(US9303033, K3, Table 12A, Compound 6)
Affinity DataIC50:  918nMpH: 7.0Assay Description:30 uM ATP: In a final reaction volume of 50 ul, recombinant PIM-1 (1 ng) was incubated with 12 mM MOPS pH 7.0, 0.4 mM EDTA, glycerol 1%, brij 35 0.00...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM218908(US9303033, O3, Table 12A, Compound 10)
Affinity DataIC50:  1.25E+3nMpH: 7.0Assay Description:30 uM ATP: In a final reaction volume of 50 ul, recombinant PIM-1 (1 ng) was incubated with 12 mM MOPS pH 7.0, 0.4 mM EDTA, glycerol 1%, brij 35 0.00...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM218906(US9303033, M3, Table 12A, Compound 8)
Affinity DataIC50:  1.45E+3nMpH: 7.0Assay Description:30 uM ATP: In a final reaction volume of 50 ul, recombinant PIM-1 (1 ng) was incubated with 12 mM MOPS pH 7.0, 0.4 mM EDTA, glycerol 1%, brij 35 0.00...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM218900(US9303033, G3, Table 12A, Compound 2)
Affinity DataIC50:  2.06E+3nMpH: 7.0Assay Description:30 uM ATP: In a final reaction volume of 50 ul, recombinant PIM-1 (1 ng) was incubated with 12 mM MOPS pH 7.0, 0.4 mM EDTA, glycerol 1%, brij 35 0.00...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM218899(US9303033, F3, Table 12A, Compound 1)
Affinity DataIC50:  2.06E+3nMpH: 7.0Assay Description:30 uM ATP: In a final reaction volume of 50 ul, recombinant PIM-1 (1 ng) was incubated with 12 mM MOPS pH 7.0, 0.4 mM EDTA, glycerol 1%, brij 35 0.00...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM218901(US9303033, H3, Table 12A, Compound 3)
Affinity DataIC50:  2.39E+3nMpH: 7.0Assay Description:30 uM ATP: In a final reaction volume of 50 ul, recombinant PIM-1 (1 ng) was incubated with 12 mM MOPS pH 7.0, 0.4 mM EDTA, glycerol 1%, brij 35 0.00...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM218907(US9303033, N3, Table 12A, Compound 9)
Affinity DataIC50: >2.50E+3nMpH: 7.0Assay Description:30 uM ATP: In a final reaction volume of 50 ul, recombinant PIM-1 (1 ng) was incubated with 12 mM MOPS pH 7.0, 0.4 mM EDTA, glycerol 1%, brij 35 0.00...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM218905(US9303033, L3, Table 12A, Compound 7)
Affinity DataIC50: >2.50E+3nMpH: 7.0Assay Description:30 uM ATP: In a final reaction volume of 50 ul, recombinant PIM-1 (1 ng) was incubated with 12 mM MOPS pH 7.0, 0.4 mM EDTA, glycerol 1%, brij 35 0.00...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM218903(US9303033, J3, Table 12A, Compound 5)
Affinity DataIC50: >2.50E+3nMpH: 7.0Assay Description:30 uM ATP: In a final reaction volume of 50 ul, recombinant PIM-1 (1 ng) was incubated with 12 mM MOPS pH 7.0, 0.4 mM EDTA, glycerol 1%, brij 35 0.00...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM218902(US9303033, I3, Table 12A, Compound 4)
Affinity DataIC50: >2.50E+3nMpH: 7.0Assay Description:30 uM ATP: In a final reaction volume of 50 ul, recombinant PIM-1 (1 ng) was incubated with 12 mM MOPS pH 7.0, 0.4 mM EDTA, glycerol 1%, brij 35 0.00...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Senhwa Biosciences

US Patent
LigandPNGBDBM218909(US9303033, P3, Table 12A, Compound 11)
Affinity DataIC50: >2.50E+3nMpH: 7.0Assay Description:30 uM ATP: In a final reaction volume of 50 ul, recombinant PIM-1 (1 ng) was incubated with 12 mM MOPS pH 7.0, 0.4 mM EDTA, glycerol 1%, brij 35 0.00...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent