Compile Data Set for Download or QSAR
maximum 50k data
Found 50 of Enz. Inhib. data with enzyme = 'Transient receptor potential cation channel subfamily V member 1' and Substrate = 'BDBM20285'
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20286(5-I-RTX | 5-iodoresiniferatoxin | [(1R,2R,6R,10S,1...)
Affinity DataKi:  0.610nM ΔG°:  -13.1kcal/mole EC50:  12.2nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20314((2R)-2-[(4-tert-butylphenyl)methyl]-3-[(2S)-2-(3-c...)
Affinity DataKi:  1.83nM ΔG°:  -12.4kcal/mole EC50:  5.20nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20311((2S)-2-[(4-tert-butylphenyl)methyl]-3-[(2S)-2-(3-c...)
Affinity DataKi:  3.29nM ΔG°:  -12.0kcal/mole EC50:  12.1nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20291(2-[(4-tert-butylphenyl)methyl]-3-[2-(3-chloro-4-me...)
Affinity DataKi:  3.60nM ΔG°:  -12.0kcal/mole EC50:  12.3nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20313((2R)-2-[(4-tert-butylphenyl)methyl]-3-[(2S)-2-(3-f...)
Affinity DataKi:  4.12nM ΔG°:  -11.9kcal/mole EC50:  0.580nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20310((2S)-2-[(4-tert-butylphenyl)methyl]-3-[(2S)-2-(3-f...)
Affinity DataKi:  6.26nM ΔG°:  -11.6kcal/mole EC50:  10.9nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20297(3-[2-(3-chloro-4-methanesulfonamidophenyl)propanam...)
Affinity DataKi:  11.3nM ΔG°:  -11.3kcal/mole EC50:  36nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20290(2-[(4-tert-butylphenyl)methyl]-3-[2-(3-fluoro-4-me...)
Affinity DataKi:  13.6nM ΔG°:  -11.2kcal/mole EC50:  3.24nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20306((2S)-2-benzyl-3-[(2S)-2-(3-fluoro-4-methanesulfona...)
Affinity DataKi:  16.5nM ΔG°:  -11.0kcal/mole EC50:  10nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20287(2-[(4-tert-butylphenyl)methyl]-3-({[(3-fluoro-4-me...)
Affinity DataKi:  22.6nM ΔG°:  -10.8kcal/mole EC50:  52nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20292(2-[(4-tert-butylphenyl)methyl]-3-[2-(4-methanesulf...)
Affinity DataKi:  24nM ΔG°:  -10.8kcal/molepH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20296(2-[(3,4-dimethylphenyl)methyl]-3-[2-(3-fluoro-4-me...)
Affinity DataKi:  33.1nM ΔG°:  -10.6kcal/mole EC50:  10.8nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20323(3-[(4-tert-butylphenyl)methyl]-1-[(1R)-1-(3-fluoro...)
Affinity DataKi:  39.2nM ΔG°:  -10.5kcal/mole EC50:  37nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20317(3-[(4-tert-butylphenyl)methyl]-1-[(1R)-1-(4-methan...)
Affinity DataKi:  41nM ΔG°:  -10.5kcal/mole EC50:  4.5nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20308((2R)-2-benzyl-3-[(2S)-2-(3-fluoro-4-methanesulfona...)
Affinity DataKi:  43nM ΔG°:  -10.4kcal/mole EC50:  8.56nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20330(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataKi:  51nM ΔG°:  -10.3kcal/molepH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20312((2R)-2-[(4-tert-butylphenyl)methyl]-3-[(2R)-2-(3-f...)
Affinity DataKi:  53nM ΔG°:  -10.3kcal/mole EC50:  30.3nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20321(3-[(4-tert-butylphenyl)methyl]-1-[(3-fluoro-4-meth...)
Affinity DataKi:  53.5nM ΔG°:  -10.3kcal/mole EC50:  9.20nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20322(3-[(4-tert-butylphenyl)methyl]-1-[1-(3-fluoro-4-me...)
Affinity DataKi:  54nM ΔG°:  -10.3kcal/mole EC50:  9.20nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20293(2-[(3,4-dimethylphenyl)methyl]-3-({[(3-fluoro-4-me...)
Affinity DataKi:  54nM ΔG°:  -10.3kcal/mole EC50:  7.80nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20289(2-[(4-tert-butylphenyl)methyl]-3-[2-(4-methanesulf...)
Affinity DataKi:  55nM ΔG°:  -10.3kcal/mole EC50:  52nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20316(3-[(4-tert-butylphenyl)methyl]-1-[1-(4-methanesulf...)
Affinity DataKi:  59.3nM ΔG°:  -10.2kcal/mole EC50:  14.7nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataKi:  63nM ΔG°:  -10.2kcal/mole EC50:  54nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20309((2S)-2-[(4-tert-butylphenyl)methyl]-3-[(2R)-2-(3-f...)
Affinity DataKi:  64nM ΔG°:  -10.2kcal/mole EC50:  142nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20331(3-[(4-tert-butylphenyl)methyl]-1-[1-(4-methanesulf...)
Affinity DataKi:  67nM ΔG°:  -10.2kcal/mole EC50:  28.6nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20298(2-[(3,4-dimethylphenyl)methyl]-3-[2-(4-methanesulf...)
Affinity DataKi:  71nM ΔG°:  -10.1kcal/mole EC50:  13.6nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20288(2-[(4-tert-butylphenyl)methyl]-3-[1-(3-fluoro-4-me...)
Affinity DataKi:  74nM ΔG°:  -10.1kcal/mole EC50:  440nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20328(3-[(4-tert-butylphenyl)methyl]-1-[(3-fluoro-4-meth...)
Affinity DataKi:  100nM ΔG°:  -9.93kcal/mole EC50:  860nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20295(2-[(3,4-dimethylphenyl)methyl]-3-[2-(4-methanesulf...)
Affinity DataKi:  119nM ΔG°:  -9.82kcal/mole EC50:  38nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20301(2-[(3,4-dimethylphenyl)methyl]-3-[2-(4-methanesulf...)
Affinity DataKi:  153nM ΔG°:  -9.66kcal/mole EC50:  133nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20294(2-[(3,4-dimethylphenyl)methyl]-3-[1-(3-fluoro-4-me...)
Affinity DataKi:  157nM ΔG°:  -9.65kcal/mole EC50:  151nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20320(1-[(4-tert-butylphenyl)methyl]-3-[1-(4-methanesulf...)
Affinity DataKi:  171nM ΔG°:  -9.60kcal/mole EC50:  60nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20325(3-[(4-tert-butylphenyl)methyl]-1-[1-(3-fluoro-4-me...)
Affinity DataKi:  230nM ΔG°:  -9.41kcal/mole EC50:  54nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20304(2-[(3,4-dimethylphenyl)methyl]-3-{[1-(4-methanesul...)
Affinity DataKi:  239nM ΔG°:  -9.39kcal/mole EC50:  118nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20300(2-[(3,4-dimethylphenyl)methyl]-3-[2-(3-fluoro-4-me...)
Affinity DataKi:  280nM ΔG°:  -9.29kcal/mole EC50:  65nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20307((2R)-2-benzyl-3-[(2R)-2-(3-fluoro-4-methanesulfona...)
Affinity DataKi:  298nM ΔG°:  -9.25kcal/mole EC50:  98nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20326(3-[(4-tert-butylphenyl)methyl]-1-[1-(3-fluoro-4-me...)
Affinity DataKi:  339nM ΔG°:  -9.18kcal/mole EC50:  223nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20299(2-[(3,4-dimethylphenyl)methyl]-3-[2-(4-methanesulf...)
Affinity DataKi:  370nM ΔG°:  -9.12kcal/mole EC50:  104nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20333(1-[(4-tert-butylphenyl)methyl]-3-[1-(4-methanesulf...)
Affinity DataKi:  370nM ΔG°:  -9.12kcal/mole EC50:  243nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20305((2S)-2-benzyl-3-[(2R)-2-(3-fluoro-4-methanesulfona...)
Affinity DataKi:  370nM ΔG°:  -9.12kcal/mole EC50:  205nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20302(2-[(3,4-dimethylphenyl)methyl]-3-{[1-(4-methanesul...)
Affinity DataKi:  396nM ΔG°:  -9.08kcal/mole EC50:  197nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20284(CHEMBL391997 | CPZ | Capsazepine | N-[2-(4-chlorop...)
Affinity DataKi:  1.30E+3nM ΔG°:  -8.35kcal/mole EC50:  520nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20284(CHEMBL391997 | CPZ | Capsazepine | N-[2-(4-chlorop...)
Affinity DataKi:  1.30E+3nM ΔG°:  -8.35kcal/mole EC50:  520nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20303(2-[(3,4-dimethylphenyl)methyl]-3-{[1-(3-fluoro-4-m...)
Affinity DataKi:  1.58E+3nM ΔG°:  -8.23kcal/mole EC50:  567nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20327(3-[(4-tert-butylphenyl)methyl]-1-[1-(3-fluoro-4-me...)
Affinity DataKi:  1.74E+3nM ΔG°:  -8.17kcal/mole EC50:  700nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20324(3-[(4-tert-butylphenyl)methyl]-1-[(1S)-1-(3-fluoro...)
Affinity DataKi:  2.14E+3nM ΔG°:  -8.04kcal/mole EC50:  2.67E+3nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20332(3-[(4-tert-butylphenyl)methyl]-1-[2-(4-methanesulf...)
Affinity DataKi:  2.89E+3nM ΔG°:  -7.86kcal/mole EC50:  663nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20318(3-[(4-tert-butylphenyl)methyl]-1-[(1S)-1-(4-methan...)
Affinity DataKi:  3.95E+3nM ΔG°:  -7.66kcal/molepH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20329(3-[(4-tert-butylphenyl)methyl]-1-[2-(3-fluoro-4-me...)
Affinity DataKi:  7.70E+3nM ΔG°:  -7.25kcal/mole EC50:  980nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

LigandPNGBDBM20319(3-[(4-tert-butylphenyl)methyl]-1-[2-(4-methanesulf...)
Affinity DataEC50:  1.80E+3nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed