TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.10E+5nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 6.92E+4nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 2.63E+4nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.74E+5nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.51E+4nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 3.55E+5nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 5.01E+3nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 1.15E+4nMAssay Description:Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 9.77E+3nMAssay Description:Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 1.17E+5nMAssay Description:Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligandMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:The compound was evaluated for pA2 at Histamine H2 receptor of guinea pig atriumMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 3.16E+4nMAssay Description:Receptor profile was evaluated at Histamine H2 receptor of guinea pig atriumMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 316nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.00E+5nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.78E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig was evaluatedMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 6.31E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 776nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 2.51E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 4.17E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 6.31E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.20E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.62E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.26E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.10E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 3.31E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 214nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 575nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.58E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 6.92E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.15E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: >5.01E+5nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 7.76E+3nMAssay Description:Potency at histamine H2 receptor subtype, was tested on guinea pig right atriumMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 3.98E+3nMAssay Description:Potency at histamine H2 receptor subtype, was tested on guinea pig right atriumMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.02E+4nMAssay Description:Potency at histamine H2 receptor subtype, was tested on guinea pig right atriumMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit
Curated by ChEMBL
Vrije Universiteit
Curated by ChEMBL
Affinity DataKd: 1.41E+4nMAssay Description:Potency at histamine H2 receptor subtype, was tested on guinea pig right atriumMore data for this Ligand-Target Pair
Affinity DataKd: 7.80E+3nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 63nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 28nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Affinity DataKd: 288nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Affinity DataKd: 562nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Affinity DataKd: 48nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Affinity DataKd: 74nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair
Affinity DataKd: 89nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair
Affinity DataKd: 120nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair