Compile Data Set for Download or QSAR
maximum 50k data
Found 106 of kd data for polymerid = 2298,2980,49000659,49000660,49000663,49000664
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50421965(CHEMBL324864)
Affinity DataKd:  1.10E+5nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKd:  6.92E+4nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM22883(CHEMBL12344 | Dimaprit | [3-(carbamimidoylsulfanyl...)
Affinity DataKd:  2.63E+4nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50421966(CHEMBL553981)
Affinity DataKd:  1.74E+5nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50421967(CHEMBL111215)
Affinity DataKd:  1.51E+4nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50421968(CHEMBL540311)
Affinity DataKd:  3.55E+5nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM22881(5-(2-aminoethyl)-4-methyl-1,3-thiazol-2-amine | Am...)
Affinity DataKd:  5.01E+3nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM22881(5-(2-aminoethyl)-4-methyl-1,3-thiazol-2-amine | Am...)
Affinity DataKd:  1.15E+4nMAssay Description:Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM22882(2-amino-5(2-aminoethyl)-4-methyl-1,3-selenazole | ...)
Affinity DataKd:  9.77E+3nMAssay Description:Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H2 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKd:  1.17E+5nMAssay Description:Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50118157(CHEMBL128635 | [1-(1-Methyl-cyclopropyl)-ethyl]-ca...)
Affinity DataKd: >1.00E+5nMAssay Description:The compound was evaluated for pA2 at Histamine H2 receptor of guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50409579(CHEMBL130005)
Affinity DataKd:  3.16E+4nMAssay Description:Receptor profile was evaluated at Histamine H2 receptor of guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405160(CHEMBL1744352)
Affinity DataKd:  316nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405161(CHEMBL555309)
Affinity DataKd:  1.00E+5nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405162(CHEMBL1626961)
Affinity DataKd:  1.78E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405163(CHEMBL541027)
Affinity DataKd:  6.31E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405164(CHEMBL1744351)
Affinity DataKd:  776nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405165(CHEMBL540256)
Affinity DataKd:  2.51E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405166(CHEMBL555668)
Affinity DataKd:  4.17E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405167(CHEMBL29770)
Affinity DataKd:  6.31E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405168(CHEMBL30946)
Affinity DataKd:  1.20E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405169(CHEMBL542087)
Affinity DataKd:  1.62E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405170(CHEMBL540005)
Affinity DataKd:  1.26E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405171(CHEMBL1744353)
Affinity DataKd:  1.10E+4nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405172(CHEMBL543520)
Affinity DataKd:  3.31E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405173(CHEMBL545393)
Affinity DataKd:  214nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405174(CHEMBL30761)
Affinity DataKd:  575nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405175(CHEMBL30578)
Affinity DataKd:  1.58E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405176(CHEMBL542817)
Affinity DataKd:  6.92E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405177(CHEMBL545625)
Affinity DataKd:  1.15E+3nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50405178(CHEMBL282769)
Affinity DataKd: >5.01E+5nMAssay Description:Antagonistic activity against H2 receptor in guinea pig.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50126902(1-[4-(4-Pyrrolidin-1-ylmethyl-benzyloxy)-phenyl]-e...)
Affinity DataKd:  7.76E+3nMAssay Description:Potency at histamine H2 receptor subtype, was tested on guinea pig right atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50126899(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)
Affinity DataKd:  3.98E+3nMAssay Description:Potency at histamine H2 receptor subtype, was tested on guinea pig right atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50126884(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)
Affinity DataKd:  1.02E+4nMAssay Description:Potency at histamine H2 receptor subtype, was tested on guinea pig right atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50126895(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-phenyl]-et...)
Affinity DataKd:  1.41E+4nMAssay Description:Potency at histamine H2 receptor subtype, was tested on guinea pig right atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50483128(Burimamide | CHEBI:3221)
Affinity DataKd:  7.80E+3nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50103506(Ranitidine | Tritec | Zantac)
Affinity DataKd:  63nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543279(CHEMBL4641916)
Affinity DataKd:  28nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543280(CHEMBL4637893)
Affinity DataKd:  14nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543281(CHEMBL4644467)
Affinity DataKd:  19nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543282(CHEMBL4645867)
Affinity DataKd:  288nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543283(CHEMBL4647775)
Affinity DataKd:  13nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543284(CHEMBL4645213)
Affinity DataKd:  562nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543285(CHEMBL4637356)
Affinity DataKd:  48nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 90 mins by flowcytometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543279(CHEMBL4641916)
Affinity DataKd:  74nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543281(CHEMBL4644467)
Affinity DataKd:  89nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543282(CHEMBL4645867)
Affinity DataKd:  120nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543283(CHEMBL4647775)
Affinity DataKd:  15nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543284(CHEMBL4645213)
Affinity DataKd:  170nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50543285(CHEMBL4637356)
Affinity DataKd:  16nMAssay Description:Binding affinity to human H2R expressed in human HEK293T cells incubated for 60 mins by automated cell imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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