Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Acetylcholinesterase' and Ligand = 'BDBM50509708'
TargetAcetylcholinesterase(Human)
Alexandria University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509708BDBM50509708(CHEMBL4458648)
Affinity DataKi:  121nMAssay Description:Mixed type inhibition of recombinant human AChE assessed as dissociation constant using acetylthiocholine iodide as substrate incubated for 10 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Alexandria University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509708BDBM50509708(CHEMBL4458648)
Affinity DataIC50: 218nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholine iodide as substrate pre-incubated for 20 mins before substrate addition and measured for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Alexandria University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509708BDBM50509708(CHEMBL4458648)
Affinity DataKi:  253nMAssay Description:Mixed type inhibition of recombinant human AChE assessed as dissociation constant for enzyme-substrate-inhibitor complex using acetylthiocholine iodi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Alexandria University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50509708BDBM50509708(CHEMBL4458648)
Affinity DataIC50: 622nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate incubated for 10 mins by spectrophotometry based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed