Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50020338
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM23840(2-[2-(2-phenylethyl)phenyl]-2,3-dihydro-1H-isoindo...)
Affinity DataIC50:  9.80E+3nMAssay Description:Antagonist activity at human recombinant LXRalpha expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activation by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM23841(2-(2-hexylphenyl)-2,3-dihydro-1H-isoindole-1,3-dio...)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at human recombinant LXRalpha expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activation by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM23840(2-[2-(2-phenylethyl)phenyl]-2,3-dihydro-1H-isoindo...)
Affinity DataIC50:  4.40E+4nMAssay Description:Antagonist activity at human recombinant LXRbeta expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activation by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM23841(2-(2-hexylphenyl)-2,3-dihydro-1H-isoindole-1,3-dio...)
Affinity DataIC50:  6.50E+4nMAssay Description:Antagonist activity at human recombinant LXRbeta expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activation by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed