Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 10556
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549563(US11306075, Ex. 7)
Affinity DataIC50:  100nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549569(US11306075, Ex. 15)
Affinity DataIC50:  100nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549574(US11306075, Ex. 21)
Affinity DataIC50:  1.17E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549558(US11306075, Ex. 2)
Affinity DataIC50:  1.27E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549564(US11306075, Ex. 8)
Affinity DataIC50:  1.31E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549560(US11306075, Ex. 4)
Affinity DataIC50:  1.39E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549576(US11306075, Ex. 23)
Affinity DataIC50:  1.57E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549570(US11306075, Ex. 16)
Affinity DataIC50:  1.93E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549568(US11306075, Ex. 14)
Affinity DataIC50:  2.06E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549579(US11306075, Ex. 28)
Affinity DataIC50:  2.48E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549561(US11306075, Ex. 5)
Affinity DataIC50:  3.03E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549575(US11306075, Ex. 22)
Affinity DataIC50:  3.42E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549577(US11306075, Ex. 24)
Affinity DataIC50:  4.02E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549567(3-[5-Bromo-3-(5-methyl-furan-2-yl)-benzofuran-2-yl...)
Affinity DataIC50:  5.78E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549566(US11306075, Ex. 12)
Affinity DataIC50:  6.09E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549562(US11306075, Ex. 6)
Affinity DataIC50:  6.35E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549559(US11306075, Ex. 3)
Affinity DataIC50:  7.55E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549571(US11306075, Ex. 18)
Affinity DataIC50:  7.67E+3nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549565(US11306075, Ex. 9)
Affinity DataIC50: >1.00E+4nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549578(US11306075, Ex. 26)
Affinity DataIC50: >1.00E+4nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549573(US11306075, Ex. 20)
Affinity DataIC50:  1.54E+4nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMicrotubule-associated protein tau(Homo sapiens (Human))
Oligomerix

US Patent
LigandPNGBDBM549572(US11306075, Ex. 19)
Affinity DataIC50:  2.08E+4nMAssay Description:Tau target (equal mixture of each construct at 300 nM) was prepared in buffer (Tris-HCl pH 7.4) and was incubated in 96-well plates at room temperatu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent