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Found 39 Enz. Inhib. hit(s) with all data for entry = 10942
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580149(US11498896, Compound 137)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580162(US11498896, Compound 211)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580132(US11498896, Compound 86)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580148(US11498896, Compound 135)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580136(US11498896, Compound 98a)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580142(US11498896, Compound 110)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580141(US11498896, Compound 106)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580146(US11498896, Compound 123)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580131(US11498896, Compound 78)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580130(US11498896, Compound 68)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580125(US11498896, Compound 27)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580161(US11498896, Compound 210)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580160(US11498896, Compound 209)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580159(US11498896, Compound 208)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580158(US11498896, Compound 206)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580157(US11498896, Compound 205)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580155(US11498896, Compound 204b)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580152(US11498896, Compound 157)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580151(US11498896, Compound 144)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580145(US11498896, Compound 122)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580143(US11498896, Compound 112)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM50518039(CHEMBL4467883 | US11498896, Compound 90)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580134(US11498896, Compound 91)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580135(US11498896, Compound 96)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580137(US11498896, Compound 99)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580140(US11498896, Compound 102a)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580154(US11498896, Compound 202b)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM50518027(CHEMBL4550815 | US11498896, Compound 1)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580124(US11498896, Compound 18b)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580147(US11498896, Compound 125)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580128(US11498896, Compound 59 | US11498896, Compound 59b)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580126(US11498896, Compound 54)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580127(US11498896, Compound 55)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580150(US11498896, Compound 140)
Affinity DataKi:  2.00E+4nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580123(US11498896, Compound 7)
Affinity DataKi:  2.00E+4nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580128(US11498896, Compound 59 | US11498896, Compound 59b)
Affinity DataKi:  2.00E+4nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM580153(US11498896, Compound 164)
Affinity DataKi:  2.00E+4nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent