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Found 21 Enz. Inhib. hit(s) with all data for entry = 11697
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640403(US20230399314, Compound 1 | US20230399314, Compoun...)
Affinity DataIC50:  4.59nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640403(US20230399314, Compound 1 | US20230399314, Compoun...)
Affinity DataIC50:  8.17nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640420(US20230399314, Compound 20)
Affinity DataIC50:  9.55nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640407(US20230399314, Compound 5)
Affinity DataIC50:  11.6nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640405(US20230399314, Compound 3)
Affinity DataIC50:  11.6nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640412(US20230399314, Compound 11)
Affinity DataIC50:  12.2nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM50552097(CHEMBL4798999 | US20230399314, Reference compound ...)
Affinity DataIC50:  12.5nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640413(US20230399314, Compound 12)
Affinity DataIC50:  15.4nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640410(US20230399314, Compound 8)
Affinity DataIC50:  16.5nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM50552106(CHEMBL4765132 | US20230399314, Reference compound ...)
Affinity DataIC50:  16.8nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640404(US20230399314, Compound 2)
Affinity DataIC50:  23.2nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640408(US20230399314, Compound 6)
Affinity DataIC50:  24.5nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM50552098(CHEMBL4792487 | US20230399314, Reference compound ...)
Affinity DataIC50:  27nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640409(US20230399314, Compound 7)
Affinity DataIC50:  32.1nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640406(US20230399314, Compound 4)
Affinity DataIC50:  58.4nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640416(US20230399314, Compound 15)
Affinity DataIC50:  123nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640418(US20230399314, Compound 17)
Affinity DataIC50:  164nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640417(US20230399314, Compound 16)
Affinity DataIC50:  173nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640419(US20230399314, Compound 19)
Affinity DataIC50:  1.25E+3nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640415(US20230399314, Compound 14)
Affinity DataIC50:  3.68E+3nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-nucleotidase(Homo sapiens (Human))
Wuhan Humanwell Innovative Drug Research and Development Center

US Patent
LigandPNGBDBM640414(US20230399314, Compound 13)
Affinity DataIC50:  6.87E+3nMAssay Description:The test was performed using Tris-MgCl2 buffer containing 25 mM Tris (Biosharp; 77-86-1) and 25 mM MgCl2 (Nanjing Chemical Reagent Co., Ltd.; 7791-18...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent