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Found 9 Enz. Inhib. hit(s) with all data for entry = 7107
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM175238(US9115082, 7)
Affinity DataKi:  9.83E+3nM IC50:  1.70E+4nMpH: 7.4Assay Description:Human recombinant adrenergic β1 receptors expressed in CHO-K1 cells are used in modified Tris-HCl buffer pH 7.4. A 25 aliquot is incubated with ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM175238(US9115082, 7)
Affinity DataKi:  2.20E+4nM IC50:  3.20E+4nMpH: 7.4Assay Description:Human recombinant adrenergic β2 receptors expressed in CHO cells are used in modified Tris-HCl buffer pH 7.4. A 50 aliquot is incubated with 0.2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM175238(US9115082, 7)
Affinity DataIC50:  1nMpH: 4.0Assay Description:The proteolytic enzyme, Dipeptidyle Peptidase IV (DppIV) was monitored in vitro by the substrate Gly-Pro 4-methoxy-β-naphthylamide while in the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50265160(1-(2-amino-2-cyclohexylacetyl)pyrrolidine-2-carbon...)
Affinity DataIC50:  46nMpH: 4.0Assay Description:The proteolytic enzyme, Dipeptidyle Peptidase IV (DppIV) was monitored in vitro by the substrate Gly-Pro 4-methoxy-β-naphthylamide while in the ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50118952(2-Amino-3-methyl-1-pyrrolidin-1-yl-butan-1-one | C...)
Affinity DataIC50:  548nMpH: 4.0Assay Description:The proteolytic enzyme, Dipeptidyle Peptidase IV (DppIV) was monitored in vitro by the substrate Gly-Pro 4-methoxy-β-naphthylamide while in the ...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50135065(2-Amino-3-methyl-1-pyrrolidin-1-yl-pentan-1-one | ...)
Affinity DataIC50:  2.00E+3nMpH: 4.0Assay Description:The proteolytic enzyme, Dipeptidyle Peptidase IV (DppIV) was monitored in vitro by the substrate Gly-Pro 4-methoxy-β-naphthylamide while in the ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM175240(US9115082, 12)
Affinity DataIC50:  8.50E+3nMpH: 4.0Assay Description:The proteolytic enzyme, Dipeptidyle Peptidase IV (DppIV) was monitored in vitro by the substrate Gly-Pro 4-methoxy-β-naphthylamide while in the ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM175239(US9115082, 11)
Affinity DataIC50:  1.20E+4nMpH: 4.0Assay Description:The proteolytic enzyme, Dipeptidyle Peptidase IV (DppIV) was monitored in vitro by the substrate Gly-Pro 4-methoxy-β-naphthylamide while in the ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM175241(US9115082, 13)
Affinity DataIC50:  3.30E+4nMpH: 4.0Assay Description:The proteolytic enzyme, Dipeptidyle Peptidase IV (DppIV) was monitored in vitro by the substrate Gly-Pro 4-methoxy-β-naphthylamide while in the ...More data for this Ligand-Target Pair
In DepthDetails US Patent